TARANABANT
Taranabant ( MK-0364) 701977-09-5 N-[3-(4-Chlorophenyl)-2(S)-(3-cyanophenyl)-1(S)-methylpropyl]-2-methyl-2-[5-(trifluoromethyl)pyridin-2-yloxy]propionamide...
View ArticlePfizer’s PF 04937319 glucokinase activators for the treatment of Type 2 diabetes
PF 04937319 N,N-dimethyl-5-(2-methyl-6-((5-methylpyrazin-2-yl)-carbamoyl)benzofuran-4-yloxy)pyrimidine-2-carboxamide MW 432.43 MF C22 H20 N6 O4 CAS 1245603-92-2 2-Pyrimidinecarboxamide,...
View ArticlePfizer’s PF 04991532 a Hepatoselective Glucokinase Activator Clinical...
PF 04991532 GKA PF-04991532 (S)-6-{3-cyclopentyl-2-[4-(trifluoromethyl)-1H-imidazol-1-yl]propanamido}nicotinic acid (S)-6-(3-Cyclopentyl-2-(4-(trifluoromethyl)-1H-imidazol-1-yl)propanamido)nicotinic...
View ArticleWO 2015177807, New patent on AVANAFIL by Wanbury
WO 2015177807 Suryakant Shivaji Pol; Nitin Sharadchandra Pradhan; Shashikant Balu Padwal; Vihar Raghunath Telange; Nitn Shankar Bondre Wanbury ltd The present invention relates to a novel compound of...
View ArticleDRL 17822 from Reddy US Therapeutics/Dr Reddy’s
CAS 920493-71-6 and CAS 898911-09-6 DRL 17822 MW 603.6045, MFC30 H31 F6 N7 Molecular Formula: C30H31F6N7 Molecular Weight: 603.604459 g/mol Cas 898911-09-6, 1454689-50-9...
View ArticleLefucoxib (乐福昔布)
Lefucoxib (乐福昔布) 5-(3,4-dimethyl-phenyl)-1-methanesulfonyl-3-trifluoromethol-pyrazole 1 [4- (methylsulfonyl) phenyl] -3-trifluoromethyl-5- (3,4-dimethylphenyl) – pyrazole CAS 849048-84-6 Molecular...
View ArticleRQ 00000010 for the treatment of GERD, functional dyspepsia and chronic...
RQ 00000010 CAS 907607-22-1 Molecular Formula: C22H27F3N2O6 Molecular Weight: 472.45479 g/mol HSMMHNBGQLGCBY-UHFFFAOYSA-N; RaQualia Pharma Inc Raqualia Pharma Inc. PFIZER INNOVATOR RQ-00000010;...
View ArticleTesmilifene , Antagonist of intracellular histamine
Tesmilifene BMS-217380; BMY-33419; DPPE CAS No. 98774-23-3(Tesmilifene), 92981-78-7(Tesmilifene hydrochloride) Tesmilifene CAS 98774-23-3 N,N-Diethyl-2-[4-(phenylmethyl)phenoxy]ethanamine DPPE...
View ArticleIptakalim Hydrochloride 盐酸埃他卡林
Iptakalim Hydrochloride 盐酸埃他卡林 NDA Filed china A K(ir) 6.1/SUR2B activator potentially for the treatment of pulmonary arterial hypertension. 179.7, C9H21N.HCl CAS No. 642407-44-1(Iptakalim)...
View ArticleZucapsaicin for osteoarthritis
Zucapsaicin (珠卡赛辛) cis-Capsaicin; (Z)-Capsaicin Zucapsaicin; Civamide; Cis-Capsaicin; 25775-90-0; (Z)-Capsaicin; (Z)-N-(4-Hydroxy-3-methoxybenzyl)-8-methylnon-6-enamide;...
View ArticleSEMAPIMOD
Semapimod Mesylate CPSI-2364, AXD-455, CN-1493, CNI 1493 CAS No. 352513-83-8(Semapimod base) Cas 164301-51-3 4x HCl CAS 872830-80-3 (Semapimod mesylate) MW 1129 CROHNS DISEASE, PHASE 1...
View ArticleWCK 5222, Wockhardt receives QIDP status for its new drug WCK 5222 from USFDA
WCK 5222 Watch this post as I get to the structure………….. DEC2015 Wockhardt has received Qualified Infectious Disease Product (QIDP) status for its new drug WCK 5222, a product from its breakthrough...
View ArticleWCK ? , WCK Series by Wockhardt for treating the bacterial infection
(2S,5R)-7-0X0-N-[(2S)-PYRROLLIDIN-2-YL-METHYLOXY]-6-(SULFOOXY)-1,6-DIAZABICYCLO[3.2.1 ]OCTANE-2-CARBOXAMIDE...
View ArticleWCK ? New molecules from Wochkardt to treat bacterial infections
(2S, 5R)-7-OXO-N-[(3S)-PYRROLIDIN-3-YLOXY]-6-(SULFOOXY)-1,6-DIAZABICYCLO [3.2.1]OCTANE-2-CARBOXAMIDE (2S,5R)-7-Oxo-N-((3S)-pyrrolidin-3-yloxy)-6-(sulfooxy)-1,6-diazabicyclo[3.2.1]octane-2-carboxamide...
View ArticleWCK ? NEW ANTIBACTERIALS FROM WOCKHARDT
WCK ? TRANS-SULFURIC ACID MONO-{2-[5-(2-METHYLAMINO-ETHYL)-[1,3,4]-OXADIAZOL-2-YL]-7-OXO-1,6-DIAZA-BICYCLO [3.2.1]OCT-6-YL} ESTER Trans-sulfuric acid mono- {...
View ArticleWCK ? trans-7-oxo-6-(sulphoxy)-1,6-diazabicvclo[3.2.1]-octane-2- carbonitrile...
. WCK ? WATCH OUT FOR THIS POST Cas 1427462-70-1 CAS 1427462-59-6, SODIUM SALT, (2S, 5R)-1,6-DIAZA-BICYCLO [3.2.1]OCTANE-2-CARBONITRILE-7-OXO-6-(SULFOOXY)-MONO SODIUM SALT Wockhardt Limited...
View ArticleFDA approves first drug to treat a rare enzyme disorder in pediatric and...
Sebelipase alfa CAS No. 1276027-63-4 Synageva… innovator ALEXION EMA AUG 28 2015 FDA approves first drug to treat a rare enzyme disorder in pediatric and adult patients 12/08/2015 Today, the U.S. Food...
View ArticleFDA approves first recombinant von Willebrand factor to treat bleeding episodes
FDA approves first recombinant von Willebrand factor to treat bleeding episodes 12/08/2015 02:44 The U.S. Food and Drug Administration today approved Vonvendi, von Willebrand factor (Recombinant), for...
View ArticleNXL104, Avibactam
NXL-104, Avibactam trans-7-oxo-6-(sulphooxy)-1,6-diazabicyclo[3,2,1]octane-2-carboxamide sodium salt (e.g., NXL-104) CAS 396731-20-7, 1192491-61-4 AVE-1330 AVE-1330A PHASE 1 a broad-spectrum...
View ArticleMK 7655, RELEBACTAM, a β-Lactamase inhibitor
MK 7655, RELEBACTAM (1R,2S,5R)-7-Oxo-N-(4-piperidinyl)-6-(sulfooxy)-1,6-diazabicyclo[3.2.1]octane-2-carboxamide (1R,2S,5R)-7-oxo-2-((piperidin-4-yl)carbamoyl)-1,6-diazabicyclo(3.2.1)octan-6-yl...
View Article